Carbajo Martínez, Rodrigo José Author

Identification of first proadrenomedullin N-terminal 20 peptide (PAMP) modulator by means of virtual screening and NMR interaction experiments

  • Roldós V.
  • Carbajo R.
  • Schott A.
  • Pineda-Lucena A.
  • Ochoa-Callejero L.
  • Martínez A.
  • Ramos A.
  • De Pascual-Teresa B.
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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY - 1/9/2012

10.1016/j.ejmech.2012.07.031

Cite count: 6 (Scopus)

How the N-terminal Domain of the OSCP Subunit of Bovine F1Fo-ATP Synthase Interacts with the N-terminal Region of an Alpha Subunit

  • Carbajo R.
  • Kellas F.
  • Yang J.
  • Runswick M.
  • Montgomery M.
  • Walker J.
  • Neuhaus D.
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Journal of Molecular Biology - 27/4/2007

10.1016/j.jmb.2007.02.059

Cite count: 27 (Scopus)
Open Access

Homologous and heterologous inhibitory effects of ATPase inhibitor proteins on F-ATPases

  • Cabezón E.
  • Jonathan G Butler P.
  • Runswick M.
  • Carbajo R.
  • Walker J.

Journal of Biological Chemistry - 1/11/2002

10.1074/jbc.m207169200

Cite count: 38 (Scopus)

Hit identification of novel heparanase inhibitors by structure- and ligand-based approaches

  • Gozalbes R.
  • Mosulén S.
  • Ortí L.
  • Rodríguez-Díaz J.
  • Carbajo R.
  • Melnyk P.
  • Pineda-Lucena A.
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BIOORGANIC and MEDICINAL CHEMISTRY - 1/4/2013

10.1016/j.bmc.2013.01.033

Cite count: 19 (Scopus)
Open Access

Glycosylation of macrolide antibiotics. Purification and kinetic studies of a macrolide glycosyltransferase from Streptomyces antibioticus

  • Quirós L.
  • Carbajo R.
  • Braña A.
  • Salas J.

Journal of Biological Chemistry - 21/4/2000

10.1074/jbc.275.16.11713

Cite count: 63 (Scopus)

Generation of potent and selective kinase inhibitors by combinatorial biosynthesis of glycosylated indolocarbazoles

  • Sánchez C.
  • Salas A.
  • Braña A.
  • Palomino M.
  • Pineda-Lucena A.
  • Carbajo R.
  • Méndez C.
  • Moris F.
  • Salas J.
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CHEMICAL COMMUNICATIONS - 10/7/2009

10.1039/b905068j

Cite count: 52 (Scopus)

Free Ligand 1D NMR Conformational Signatures to Enhance Structure Based Drug Design of a Mcl-1 Inhibitor (AZD5991) and Other Synthetic Macrocycles

  • Balazs A.
  • Carbajo R.
  • Davies N.
  • Dong Y.
  • Hird A.
  • Johannes J.
  • Lamb M.
  • McCoull W.
  • Raubo P.
  • Robb G.
  • Packer M.
  • Chiarparin E.
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JOURNAL OF MEDICINAL CHEMISTRY - 14/11/2019

10.1021/acs.jmedchem.9b00716

Cite count: 16 (Scopus)

Diversity-orientated synthesis of macrocyclic heterocycles using a double SNAr approach

  • Raubo P.
  • Carbajo R.J.
  • McCoull W.
  • Raubo J.
  • Thomas M.

ORGANIC and BIOMOLECULAR CHEMISTRY - 28/7/2021

10.1039/d1ob00612f

Cite count:

Discovery of Pyrazolo[1,5-a]pyrimidine B-Cell Lymphoma 6 (BCL6) Binders and Optimization to High Affinity Macrocyclic Inhibitors

  • McCoull W.
  • Abrams R.
  • Anderson E.
  • Blades K.
  • Barton P.
  • Box M.
  • Burgess J.
  • Byth K.
  • Cao Q.
  • Chuaqui C.
  • Carbajo R.
  • Cheung T.
  • Code E.
  • Ferguson A.
  • Fillery S.
  • Fuller N.
  • Gangl E.
  • Gao N.
  • Grist M.
  • Hargreaves D.
  • Howard M.
  • Hu J.
  • Kemmitt P.
  • Nelson J.
  • O’Connell N.
  • Prince D.
  • Raubo P.
  • Rawlins P.
  • Robb G.
  • Shi J.
  • Waring M.
  • Whittaker D.
  • Wylot M.
  • Zhu X.
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JOURNAL OF MEDICINAL CHEMISTRY - 25/5/2017

10.1021/acs.jmedchem.7b00359

Cite count: 38 (Scopus)

Discovery of AZD9833, a Potent and Orally Bioavailable Selective Estrogen Receptor Degrader and Antagonist

  • Scott J.S.
  • Moss T.A.
  • Balazs A.
  • Barlaam B.
  • Breed J.
  • Carbajo R.J.
  • Chiarparin E.
  • Davey P.R.J.
  • Delpuech O.
  • Fawell S.
  • Fisher D.I.
  • Gagrica S.
  • Gangl E.T.
  • Grebe T.
  • Greenwood R.D.
  • Hande S.
  • Hatoum-Mokdad H.
  • Herlihy K.
  • Hughes S.
  • Hunt T.A.
  • Huynh H.
  • Janbon S.L.M.
  • Johnson T.
  • Kavanagh S.
  • Klinowska T.
  • Lawson M.
  • Lister A.S.
  • Marden S.
  • McGinnity D.F.
  • Morrow C.J.
  • Nissink J.W.M.
  • O'Donovan D.H.
  • Peng B.
  • Polanski R.
  • Stead D.S.
  • Stokes S.
  • Thakur K.
  • Throner S.R.
  • Tucker M.J.
  • Varnes J.
  • Wang H.
  • Wilson D.M.
  • Wu D.
  • Wu Y.
  • Yang B.
  • Yang W.
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JOURNAL OF MEDICINAL CHEMISTRY - 10/12/2020

10.1021/acs.jmedchem.0c01163

Cite count: 8 (Scopus)

Aplicación de métodos de rmn de detección inversa a través de 1h y 31p a la identificación de moléculas complejas y núcleos de gamma baja

  • Rodrigo José Carbajo Martínez
  • Fernando Lopez-Ortiz

1999

Cite count:
  • Dialnet

This author has no conferences.

This author has no patents.

Erratum: Free ligand 1D NMR conformational signatures to enhance structure based drug design of a Mcl-1 inhibitor (AZD5991) and other synthetic macrocycles (Journal of Medicinal Chemistry (2019) 62:21 (9418-9437) DOI: 10.1021/acs.jmedchem.9b00716)

  • Balazs A.Y.S.
  • Carbajo R.J.
  • Davies N.L.
  • Dong Y.
  • Hird A.W.
  • Johannes J.W.
  • Lamb M.L.
  • McCoull W.
  • Raubo P.
  • Robb G.R.
  • Packer M.J.
  • Chiarparin E.
... View more Collapse

JOURNAL OF MEDICINAL CHEMISTRY - 1/1/2021

10.1021/acs.jmedchem.1c00273

Cite count:

Scopus: 24

Web of Science: 5

Scopus: 47

Web of Science: 4

Last data update: 5/18/24 6:26 AM
Next scheduled update: 5/25/24 3:00 AM