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Carbajo Martínez, Rodrigo José Author

Structure-Activity Relationship of Oxacyclo- and Triazolo-Containing Respiratory Syncytial Virus Polymerase Inhibitors

  • Tran M.T.
  • Grosse S.
  • Carbajo R.J.
  • Jacoby E.
  • Yin Y.
  • Yu X.
  • Martinez C.
  • Stoops B.
  • Cooymans L.
  • Hu L.
  • Lutter F.H.
  • Pieters S.
  • Tan E.
  • Alcázar J.
  • Roymans D.
  • van Vlijmen H.
  • Rigaux P.
  • Sharma S.
  • Jonckers T.H.M.
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ACS Medicinal Chemistry Letters - 12/9/2024

10.1021/acsmedchemlett.4c00272

Cite count:

Synthesis of polysubstituted azepanes by dearomative ring expansion of nitroarenes

  • Mykura R.
  • Sánchez-Bento R.
  • Matador E.
  • Duong V.K.
  • Varela A.
  • Angelini L.
  • Carbajo R.J.
  • Llaveria J.
  • Ruffoni A.
  • Leonori D.
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Nature Chemistry - 1/5/2024

10.1038/s41557-023-01429-1

Cite count: 15 (Scopus)
  • CiteScore: 29.6 (2023)
  • SJR: 6.94 (2023
  • SNIP: 3.334 (2023
Open Access

Metabolism-driven in vitro/in vivo disconnect of an oral ERɑ VHL-PROTAC

  • Hayhow T.G.
  • Williamson B.
  • Lawson M.
  • Cureton N.
  • Braybrooke E.L.
  • Campbell A.
  • Carbajo R.J.
  • Cheraghchi-Bashi A.
  • Chiarparin E.
  • Diène C.R.
  • Fallan C.
  • Fisher D.I.
  • Goldberg F.W.
  • Hopcroft L.
  • Hopcroft P.
  • Jackson A.
  • Kettle J.G.
  • Klinowska T.
  • Künzel U.
  • Lamont G.
  • Lewis H.J.
  • Maglennon G.
  • Martin S.
  • Gutierrez P.M.
  • Morrow C.J.
  • Nikolaou M.
  • Nissink J.W.M.
  • O’Shea P.
  • Polanski R.
  • Schade M.
  • Scott J.S.
  • Smith A.
  • Weber J.
  • Wilson J.
  • Yang B.
  • Crafter C.
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Communications Biology - 1/12/2024

10.1038/s42003-024-06238-x

Cite count:

Design of rigid protein-protein interaction inhibitors enables targeting of undruggable Mcl-1

  • Hargreaves D.
  • Carbajo R.J.
  • Bodnarchuk M.S.
  • Embrey K.
  • Rawlins P.B.
  • Packer M.
  • Degorce S.L.
  • Hird A.W.
  • Johannes J.W.
  • Chiarparin E.
  • Schade M.
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PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA - 23/5/2023

10.1073/pnas.2221967120

Cite count:
  • JCR Impact Factor: 9.4 (2023)
  • CiteScore: 19.2 (2022)
  • SJR: 4.026 (2022
  • SNIP: 2.765 (2022
  • JCR 5-year Impact Factor: 10.8
  • JCR Categories: MULTIDISCIPLINARY SCIENCES

Discovery of a Potent and Orally Bioavailable Zwitterionic Series of Selective Estrogen Receptor Degrader-Antagonists

  • Scott J.S.
  • Stead D.
  • Barlaam B.
  • Breed J.
  • Carbajo R.J.
  • Chiarparin E.
  • Cureton N.
  • Davey P.R.J.
  • Fisher D.I.
  • Gangl E.T.
  • Grebe T.
  • Greenwood R.D.
  • Hande S.
  • Hatoum-Mokdad H.
  • Hughes S.J.
  • Hunt T.A.
  • Johnson T.
  • Kavanagh S.L.
  • Klinowska T.C.M.
  • Larner C.J.B.
  • Lawson M.
  • Lister A.S.
  • Longmire D.
  • Marden S.
  • McGuire T.M.
  • McMillan C.
  • McMurray L.
  • Morrow C.J.
  • Nissink J.W.M.
  • Moss T.A.
  • O’Donovan D.H.
  • Polanski R.
  • Stokes S.
  • Thakur K.
  • Trueman D.
  • Truman C.
  • Tucker M.J.
  • Wang H.
  • Whalley N.
  • Wu D.
  • Wu Y.
  • Yang B.
  • Yang W.
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JOURNAL OF MEDICINAL CHEMISTRY - 23/2/2023

10.1021/acs.jmedchem.2c01964

Cite count: 5 (Scopus)
  • JCR Impact Factor: 6.8 (2023)
  • CiteScore: 12.3 (2022)
  • SJR: 1.805 (2022
  • SNIP: 1.655 (2022
  • JCR 5-year Impact Factor: 7.1
  • JCR Categories: CHEMISTRY, MEDICINAL

Structural and mechanistic insights into the inhibition of respiratory syncytial virus polymerase by a non-nucleoside inhibitor

  • Yu X.
  • Abeywickrema P.
  • Bonneux B.
  • Behera I.
  • Anson B.
  • Jacoby E.
  • Fung A.
  • Adhikary S.
  • Bhaumik A.
  • Carbajo R.J.
  • De Bruyn S.
  • Miller R.
  • Patrick A.
  • Pham Q.
  • Piassek M.
  • Verheyen N.
  • Shareef A.
  • Sutto-Ortiz P.
  • Ysebaert N.
  • Van Vlijmen H.
  • Jonckers T.H.M.
  • Herschke F.
  • McLellan J.S.
  • Decroly E.
  • Fearns R.
  • Grosse S.
  • Roymans D.
  • Sharma S.
  • Rigaux P.
  • Jin Z.
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Communications Biology - 1/12/2023

10.1038/s42003-023-05451-4

Cite count:
  • JCR Impact Factor: 5.2 (2023)
  • JCR 5-year Impact Factor: 5.6
  • JCR Categories: BIOLOGY

Relating Conformational Equilibria to Conformer-Specific Lipophilicities: New Opportunities in Drug Discovery

  • Linclau B.
  • Wang Z.
  • Jeffries B.
  • Graton J.
  • Carbajo R.J.
  • Sinnaeve D.
  • Le Questel J.Y.
  • Scott J.S.
  • Chiarparin E.
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ANGEWANDTE CHEMIE-INTERNATIONAL EDITION - 7/2/2022

10.1002/anie.202114862

Cite count: 4 (Scopus)
  • JCR Impact Factor: 16.6 (2022)
  • CiteScore: 23.9 (2021)
  • SJR: 5.126 (2021
  • SNIP: 2.323 (2021
  • JCR 5-year Impact Factor: 15.3
  • JCR Categories: CHEMISTRY, MULTIDISCIPLINARY

Structure of human spermine oxidase in complex with a highly selective allosteric inhibitor

  • Diaz E.
  • Adhikary S.
  • Tepper A.W.J.W.
  • Riley D.
  • Ortiz-Meoz R.
  • Krosky D.
  • Buyck C.
  • Lamenca C.M.
  • Llaveria J.
  • Fang L.
  • Kalin J.H.
  • Klaren V.N.A.
  • Fahmy S.
  • Shaffer P.L.
  • Kirkpatrick R.
  • Carbajo R.J.
  • Thomsen M.
  • Impagliazzo A.
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Communications Biology - 1/12/2022

10.1038/s42003-022-03735-9

Cite count:
  • JCR Impact Factor: 5.9 (2022)
  • JCR 5-year Impact Factor: 6.3
  • JCR Categories: BIOLOGY

Impact of PROTAC Linker Plasticity on the Solution Conformations and Dissociation of the Ternary Complex

  • Weerakoon D.
  • Carbajo R.J.
  • De Maria L.
  • Tyrchan C.
  • Zhao H.

Journal of Chemical Information and Modeling - 24/1/2022

10.1021/acs.jcim.1c01036

Cite count: 6 (Scopus)
  • JCR Impact Factor: 5.6 (2022)
  • CiteScore: 7.7 (2021)
  • SJR: 1.223 (2021
  • SNIP: 1.339 (2021
  • JCR 5-year Impact Factor: 5.9
  • JCR Categories: COMPUTER SCIENCE, INTERDISCIPLINARY APPLICATIONS

Discovery of AZD4625, a Covalent Allosteric Inhibitor of the Mutant GTPase KRASG12C

  • Kettle J.G.
  • Bagal S.K.
  • Bickerton S.
  • Bodnarchuk M.S.
  • Boyd S.
  • Breed J.
  • Carbajo R.J.
  • Cassar D.J.
  • Chakraborty A.
  • Cosulich S.
  • Cumming I.
  • Davies M.
  • Davies N.L.
  • Eatherton A.
  • Evans L.
  • Feron L.
  • Fillery S.
  • Gleave E.S.
  • Goldberg F.W.
  • Hanson L.
  • Harlfinger S.
  • Howard M.
  • Howells R.
  • Jackson A.
  • Kemmitt P.
  • Lamont G.
  • Lamont S.
  • Lewis H.J.
  • Liu L.
  • Niedbala M.J.
  • Phillips C.
  • Polanski R.
  • Raubo P.
  • Robb G.
  • Robinson D.M.
  • Ross S.
  • Sanders M.G.
  • Tonge M.
  • Whiteley R.
  • Wilkinson S.
  • Yang J.
  • Zhang W.
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JOURNAL OF MEDICINAL CHEMISTRY - 1/1/2022

10.1021/acs.jmedchem.2c00369

Cite count: 10 (Scopus)
  • JCR Impact Factor: 7.3 (2022)
  • CiteScore: 11.5 (2021)
  • SJR: 1.888 (2021
  • SNIP: 1.841 (2021
  • JCR 5-year Impact Factor: 7.3
  • JCR Categories: CHEMISTRY, MEDICINAL

Aplicación de métodos de rmn de detección inversa a través de 1h y 31p a la identificación de moléculas complejas y núcleos de gamma baja

  • Rodrigo José Carbajo Martínez
  • Fernando Lopez-Ortiz

1999

Cite count:
  • Dialnet

This author has no conferences.

This author has no patents.

Erratum: Free ligand 1D NMR conformational signatures to enhance structure based drug design of a Mcl-1 inhibitor (AZD5991) and other synthetic macrocycles (Journal of Medicinal Chemistry (2019) 62:21 (9418-9437) DOI: 10.1021/acs.jmedchem.9b00716)

  • Balazs A.Y.S.
  • Carbajo R.J.
  • Davies N.L.
  • Dong Y.
  • Hird A.W.
  • Johannes J.W.
  • Lamb M.L.
  • McCoull W.
  • Raubo P.
  • Robb G.R.
  • Packer M.J.
  • Chiarparin E.
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JOURNAL OF MEDICINAL CHEMISTRY - 1/1/2021

10.1021/acs.jmedchem.1c00273

Cite count:
  • JCR Impact Factor: 8.039 (2021)
  • CiteScore: 10.6 (2020)
  • SJR: 2.01 (2020
  • SNIP: 1.791 (2020
  • JCR 5-year Impact Factor: 7.897
  • JCR Categories: CHEMISTRY, MEDICINAL

Scopus: 24

Web of Science: 5

Scopus: 48

Web of Science: 4

Last data update: 11/23/24 6:59 AM
Next scheduled update: 11/30/24 3:00 AM